Azilsartan

Azilsartan (CAS 147403-03-0), also referenced under the development code TAK-536, is an angiotensin II receptor blocker (ARB) active pharmaceutical ingredient used in the treatment of hypertension.

Where is Azilsartan used?

• Pharmaceutical manufacturing: core active ingredient for antihypertensive tablet formulations
• CDMOs: reference standard or synthetic intermediate for generic equivalents of branded ARB products
• Analytical and QA workflows: characterized API material for regulatory submissions of generic antihypertensive drugs
• Research institutions procure it for pharmacological studies comparing ARB receptor selectivity and binding profiles.

Good to know: It serves as the free acid form of the prodrug azilsartan medoxomil.

Commercial specifications

• Offered at research, pilot, and commercial scale